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Pain Research
TRPV1 Channel Related Products

Transient receptor potential vanilloid 1 (TRPV1) is one of the TRP channels cloned as a capsaicin receptor, functions as a pain receptor, and is activated by capsaicin, heat, and protons.

INDEX

  1. New Products
    AMG9810
    2-APB
    BCTC     NEW
    Capsazepine
    Olvanil     NEW
    SB-366791
  2. Product List
  3. Related Products


1. New Products

AMG9810

AMG9810 is an antagonist of transient receptor potential vanilloid 1 (TRPV1).
It also inhibits the activation of TRPV1 by heat and protons, besides capsaicin.

  • Appearance: White - brown, Crystals - powder
  • Assay (HPLC): 98.0+ %
  • Solubility in ethanol: to pass test
  • CAS No.: 545395-94-6
  • C21H23NO3 = 337.41

AMG9810
2-APB

2-Aminoethoxydiphenyl borate (2APB) can block TRP channels TRPC1, TRPC3, TRPC5, TRPC6, TRPV6, TRPM3, TRPM7, TRPM8 and TRPP2. At high concentrations 2-APB can activate TRPV1, TRPV2 and TRPV3. It is also an inhibitor of inositol triphosphate (IP3) receptors.

  • Appearance: White - brown, Crystalline powder - powder
  • Assay (HPLC): 98.0+ %
  • Solubility in ethanol: to pass test.
  • CAS No.:524-95-8
  • C14H16BNO = 225.09

2-APB
BCTC

BCTC is an antagonist of transient receptor potential vanilloid 1 (TRPV1). TRPV1 is one of the TRP channels cloned as a capsaicin receptor, functions as a pain receptor, and is activated by capsaicin, heat, and protons. BCTC inhibits the activation of TRPV1 by capsaicin and acids.

  • Appearance: White - pale brown, Crystalline powder - powder
  • Assay (HPLC): 98.0+ %
  • Solubility in ethanol: to pass test.
  • CAS No.:393514-24-4
  • C20H25ClN4O = 372.89
BCTC
Capsazepine

Capsazepine is an analog of capsaicin, and an antagonist of transient receptor potential vanilloid 1 (TRPV1).

  • Appearance: White - pale yellow, Crystalline powder - powder or mass
  • Assay (HPLC): 98.0+ %
  • Solubility in ethanol: to pass test.
  • CAS No.:138977-28-3
  • C19H21ClN2O2S = 376.90
Capsazepine
Olvanil

Olvanil is a potent antagonist of transient receptor potential vanilloid 1 (TRPV1). It also acts as an agonist for CB1.

  • Appearance: White - pale yellow, Crystalline powder - powder
  • Assay (HPLC): 98.0+ %
  • Solubility in ethanol: to pass test.
  • CAS No.:58493-49-5
  • C26H43NO3 = 417.62
Olvanil
SB-366791

SB-366791 is an antagonist of transient receptor potential vanilloid 1 (TRPV1). It inhibits the activation of TRPV1 by capsaicin and heat. It has been reported that it does not inhibit activation by protons.

  • Appearance: White - pale brown, Crystals - powder
  • Assay (HPLC): 98.0+ %
  • Solubility in ethanol: to pass test.
  • CAS No.:472981-92-3
  • C16H14ClNO2 = 287.74


SB-366791

2.Producrt List

Product Name Pkg. Size Wako Cat. No. Grade Storage Condition
AMG9810 10 mg 015-25071 for Cellbiology Keep at 2 - 10°C.
50 mg 011-25073
2-APB 100 mg 013-24911 Keep at -20°C.
500 mg 019-24913
BCTC 10 mg 027-18241
50 mg 023-18243
Capsazepine 10 mg 037-23171
50 mg 033-23173
Olvanil 10 mg 154-03231
50 mg 150-03233
SB-366791 10 mg 193-17431
50 mg 199-17433



3. Related Products

Product Name Pkg. Size Wako Cat. No. Grade/
Manufacturer's code
Storage Condition
TRPV1 Agonist
Capsaicin 100 mg 034-11351 Wako 1st Grade Keep at 2 - 10°C.
1 g 030-11353
TRPV1 Antagonist
Ruthenium Red 100 mg 184-00331 Wako Special Grade Keep at room temperature.
1 g 180-00333
TRPV1 Antibodies
Anti Rat TRPV1(VR-1) Polyclonal Antibody, Rabbit 5 μg 300-08991 TransGenic Inc.
KM018
Keep at -20°C.
Anti Rat phospho TRPV1(VR-1) Polyclonal Antibody 25 μg 301-31871 TransGenic Inc.
KM112
Keep at -20°C.
QUOTATION REQUEST
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